TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Shinshu University
Curated by PDSP Ki Database
Shinshu University
Curated by PDSP Ki Database
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Shinshu University
Curated by PDSP Ki Database
Shinshu University
Curated by PDSP Ki Database
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Shinshu University
Curated by PDSP Ki Database
Shinshu University
Curated by PDSP Ki Database
Affinity DataKi: 2.60E+3nMAssay Description:Competitive inhibition of recombinant human Cdc25B (351 to 380 residues) assessed as hydrolysis of substrate O-methylfluorescein phosphate by Linewea...More data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Shinshu University
Curated by ChEMBL
Shinshu University
Curated by ChEMBL
Affinity DataIC50: 530nMAssay Description:Inhibition of FLAG-tagged full-length human recombinant DYRK1A (127 to 485 residues) expressed in Escherichia coli assessed as reduction in autophosp...More data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Shinshu University
Curated by ChEMBL
Shinshu University
Curated by ChEMBL
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of FLAG-tagged full-length human recombinant DYRK1A (127 to 485 residues) expressed in Escherichia coli assessed as reduction in autophosp...More data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Shinshu University
Curated by ChEMBL
Shinshu University
Curated by ChEMBL
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of FLAG-tagged full-length human recombinant DYRK1A (127 to 485 residues) expressed in Escherichia coli assessed as reduction in autophosp...More data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Shinshu University
Curated by ChEMBL
Shinshu University
Curated by ChEMBL
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of FLAG-tagged full-length human recombinant DYRK1A (127 to 485 residues) expressed in Escherichia coli assessed as reduction in autophosp...More data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Shinshu University
Curated by ChEMBL
Shinshu University
Curated by ChEMBL
Affinity DataIC50: 4.50E+3nMAssay Description:Inhibition of FLAG-tagged full-length human recombinant DYRK1A (127 to 485 residues) expressed in Escherichia coli assessed as reduction in autophosp...More data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Shinshu University
Curated by ChEMBL
Shinshu University
Curated by ChEMBL
Affinity DataIC50: 4.50E+3nMAssay Description:Inhibition of FLAG-tagged full-length human recombinant DYRK1A (127 to 485 residues) expressed in Escherichia coli assessed as reduction in autophosp...More data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Shinshu University
Curated by ChEMBL
Shinshu University
Curated by ChEMBL
Affinity DataIC50: 7.40E+3nMAssay Description:Inhibition of FLAG-tagged full-length human recombinant DYRK1A (127 to 485 residues) expressed in Escherichia coli assessed as reduction in autophosp...More data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Shinshu University
Curated by ChEMBL
Shinshu University
Curated by ChEMBL
Affinity DataIC50: 1.30E+4nMAssay Description:Inhibition of FLAG-tagged full-length human recombinant DYRK1A (127 to 485 residues) expressed in Escherichia coli assessed as reduction in autophosp...More data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Shinshu University
Curated by ChEMBL
Shinshu University
Curated by ChEMBL
Affinity DataIC50: >3.20E+4nMAssay Description:Inhibition of FLAG-tagged full-length human recombinant DYRK1A (127 to 485 residues) expressed in Escherichia coli assessed as reduction in autophosp...More data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Shinshu University
Curated by ChEMBL
Shinshu University
Curated by ChEMBL
Affinity DataIC50: >3.20E+4nMAssay Description:Inhibition of FLAG-tagged full-length human recombinant DYRK1A (127 to 485 residues) expressed in Escherichia coli assessed as reduction in autophosp...More data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Shinshu University
Curated by ChEMBL
Shinshu University
Curated by ChEMBL
Affinity DataIC50: >3.20E+4nMAssay Description:Inhibition of FLAG-tagged full-length human recombinant DYRK1A (127 to 485 residues) expressed in Escherichia coli assessed as reduction in autophosp...More data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Shinshu University
Curated by ChEMBL
Shinshu University
Curated by ChEMBL
Affinity DataIC50: 3.50E+4nMAssay Description:Inhibition of FLAG-tagged full-length human recombinant DYRK1A (127 to 485 residues) expressed in Escherichia coli assessed as reduction in autophosp...More data for this Ligand-Target Pair
Affinity DataIC50: 2.08E+5nMAssay Description:Inhibition of mushroom tyrosinaseMore data for this Ligand-Target Pair
Affinity DataIC50: 2.89E+5nMAssay Description:Inhibition of mushroom tyrosinaseMore data for this Ligand-Target Pair
Affinity DataIC50: 4.90E+5nMAssay Description:Inhibition of mushroom tyrosinaseMore data for this Ligand-Target Pair